SCHEMBL3417280

SCHEMBL3417280

COc1ccc(F)cc1C(Br)C=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.40
NFE2L2 Q16236 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40
HTT P42858 2/20 0.39
KDM4E B2RXH2 2/20 0.38
PTGS1 P23219 1/20 0.37
TSHR P16473 2/20 0.37
ALK Q9UM73 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5786635 0.87 KDM4E (0.38) ERN1NFE2L2ALDH1A1MEN1POLB
SCHEMBL20486787 0.83 KDM4E (0.41) ERN1NFE2L2ALDH1A1MEN1POLB
SCHEMBL3641536 0.81 HTT (0.40) ERN1ALDH1A1MEN1KMT2AHTT
SCHEMBL3411434 0.81 ACHE (0.47) ERN1ALDH1A1MEN1POLBHPGD
SCHEMBL28963070 0.81 HTT (0.58) ALDH1A1MEN1KMT2AHTTTSHR
SCHEMBL2928368 0.81 HTT (0.58) ALDH1A1MEN1KMT2AHTTTSHR
SCHEMBL169082 0.80 CA1 (0.46) ERN1NFE2L2ALDH1A1MEN1POLB
SCHEMBL16794847 0.80 ERN1 (0.40) ERN1NFE2L2ALDH1A1POLBHTT
SCHEMBL3637979 0.80 ALDH1A1 (0.40) ERN1ALDH1A1MEN1POLBHPGD
SCHEMBL27869432 0.79 NFE2L2 (0.41) NFE2L2MEN1KMT2AKDM4EPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018161008-A1 PROCESSES FOR THE PREPARATION OF FUNGICIDAL COMPOUNDS GILEAD APOLLO, LLC (US) 2018-09-07 WO disclosed
EP-2265606-A1 HEPATITIS C VIRUS INHIBITORS Bristol-Myers Squibb Company (US) 2010-12-29 EP disclosed
WO-2009129109-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-10-22 WO disclosed
EP-1583742-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-12 EP disclosed
WO-2004060870-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-22 WO disclosed