SCHEMBL16795392

SCHEMBL16795392

CN1CCCN(Cc2cc(B3OC(C)(C)C(C)(C)O3)ccc2O)CC1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
ACHE P22303 2/20 0.42
CACNA1B Q00975 1/20 0.41
TSHR P16473 1/20 0.41
GFER P55789 1/20 0.41
CHKA P35790 4/20 0.40
NR1D1 P20393 1/20 0.40
NR1D2 Q14995 1/20 0.40
CA2 P00918 1/20 0.39
NCF1 P14598 1/20 0.39
PRMT6 Q96LA8 1/20 0.39
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16795211 0.91 POLB (0.46) KDM4EALDH1A1POLBTDP1ACHE
SCHEMBL16795161 0.84 POLB (0.42) KDM4EALDH1A1POLBTDP1CHKA
SCHEMBL16795319 0.82 POLB (0.44) KDM4EALDH1A1POLBTDP1CHKA
SCHEMBL16121847 0.80 CHKA (0.60) KDM4ECHKACA2NCF1PRMT6
SCHEMBL21565713 0.79 ALDH1A1 (0.42) KDM4EALDH1A1POLBTDP1CHKA
SCHEMBL29725194 0.79 ALDH1A1 (0.42) KDM4EALDH1A1POLBTDP1CHKA
SCHEMBL16795274 0.78 PARP1 (0.38) KDM4EALDH1A1POLBACHECACNA1B
SCHEMBL18579955 0.78 ROCK1 (0.53) KDM4EALDH1A1POLBTDP1CHKA
SCHEMBL34461817 0.75 ALDH1A1 (0.44) KDM4EALDH1A1
SCHEMBL16795175 0.75 KDM4E (0.70) KDM4EALDH1A1POLBTDP1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed