SCHEMBL16795274

SCHEMBL16795274

CN(C)C1CCN(Cc2cc(B3OC(C)(C)C(C)(C)O3)ccc2O)CC1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.38
HIF1A Q16665 4/20 0.36
ACHE P22303 2/20 0.36
CACNA1B Q00975 1/20 0.36
CTSB P07858 1/20 0.36
TSHR P16473 1/20 0.35
GFER P55789 1/20 0.35
BACE1 P56817 1/20 0.35
ROCK1 Q13464 1/20 0.35
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
POLB P06746 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
TNKS O95271 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18580822 0.78 MAPT (0.39) ACHETSHRKDM4EALDH1A1POLB
SCHEMBL16795392 0.78 KDM4E (0.43) ACHECACNA1BTSHRGFERBACE1
SCHEMBL27159868 0.77 KDM4E (0.47) HIF1AROCK1KDM4EALDH1A1POLB
SCHEMBL16826595 0.77 PARP1 (0.39) PARP1KDM4EALDH1A1TNKS
SCHEMBL16795302 0.75 ALDH1A1 (0.54) HIF1ATSHRKDM4EALDH1A1SMN1; SMN2
SCHEMBL16858885 0.75 ROCK1 (0.48) ACHEBACE1ROCK1ALDH1A1
SCHEMBL18580094 0.74 LTA4H (0.49) PARP1
SCHEMBL18580092 0.74 LTA4H (0.49) PARP1
SCHEMBL18580625 0.74 LTA4H (0.49) PARP1
SCHEMBL18580722 0.73 LPL (0.45) PARP1KDM4ETNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015086693-A1 PYRAZOLOPYRIMIDIN-2-YL DERIVATIVES AS JAK INHIBITORS ALMIRALL, S.A. (ES) 2015-06-18 WO disclosed