SCHEMBL16795470

SCHEMBL16795470

CC(=O)c1cccnc1.CN(C)/C=C/C(=O)c1cccnc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.58
RECQL P46063 2/20 0.57
MAPT P10636 6/20 0.56
KMT2A Q03164 2/20 0.56
MEN1 O00255 1/20 0.56
CYP1A1 P04798 3/20 0.52
CYP1A2 P05177 3/20 0.52
CYP1B1 Q16678 3/20 0.52
CYP3A4 P08684 2/20 0.52
CYP2D6 P10635 2/20 0.52
MAPK1 P28482 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
GAA P10253 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HPGD P15428 2/20 0.49
LMNA P02545 3/20 0.48
GPR52 Q9Y2T5 1/20 0.47
APP P05067 1/20 0.47
GSK3B P49841 1/20 0.47
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6258932 1.00 HTT (0.58) HTTRECQLMAPTKMT2AMEN1
SCHEMBL1218 0.94 HTT (0.65) HTTRECQLMAPTKMT2AMEN1
SCHEMBL1643 0.94 HTT (0.65) HTTRECQLMAPTKMT2AMEN1
SCHEMBL30269691 0.94 HTT (0.65) HTTRECQLMAPTKMT2AMEN1
SCHEMBL29364482 0.94 HTT (0.65) HTTRECQLMAPTKMT2AMEN1
SCHEMBL9486033 0.94 HTT (0.65) HTTRECQLMAPTKMT2AMEN1
SCHEMBL29496911 0.80
SCHEMBL1699 0.80
SCHEMBL8039612 0.80
Hydrochloric Acid SCHEMBL4897791 0.79 ALDH1A1 (0.63) HTTKMT2ACYP1A2CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015087343-A2 AN IMPROVED PROCESS FOR THE PREPARATION OF NILOTINIB AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF LAURUS LABS PRIVATE LIMITED (IN) 2015-06-18 WO disclosed