SCHEMBL16796019

SCHEMBL16796019

O=C(c1ccccc1)c1ccccc1C#Cc1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.48
GAA P10253 3/20 0.46
MAPT P10636 1/20 0.46
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
ALDH1A1 P00352 4/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
MAPK14 Q16539 1/20 0.41
IKBKB O14920 1/20 0.41
ALOX15 P16050 1/20 0.40
CNR2 P34972 1/20 0.40
ATM Q13315 2/20 0.40
CDC25B P30305 1/20 0.40
HSP90AA1 P07900 1/20 0.39
PKM P14618 1/20 0.39
CCR6 P51684 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TLR9 Q9NR96 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29855934 0.82 NPC1 (0.66) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL4444737 0.82 NPC1 (0.66) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL16796021 0.82 NPC1 (0.53) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL333008 0.79 AKR1C3 (0.61) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL29433447 0.79 AKR1C3 (0.61) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL4300998 0.79 NPC1 (0.57) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL31317034 0.79 NPC1 (0.66) GAAMAPTNPC1RAB9AALDH1A1
SCHEMBL16796015 0.79 CA12 (0.51) AKR1C3GAAMAPTNPC1RAB9A
SCHEMBL64069 0.76 AKR1C3 (0.57) AKR1C3GAAMAPTALDH1A1ATM
SCHEMBL1331831 0.76 AKR1C3 (0.57) AKR1C3GAAMAPTALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080189-B1 POLYMERIC MATERIALS VICTREX MFG LTD (GB) 2020-02-12 EP disclosed
US-20160304667-A1 POLYMERIC MATERIALS VICTREX MANUFACTURING LIMITED (GB) 2016-10-20 US disclosed
EP-3080189-A1 POLYMERIC MATERIALS Victrex Manufacturing Limited (GB) 2016-10-19 EP disclosed
WO-2015087059-A1 POLYMERIC MATERIALS VICTREX MANUFACTURING LIMITED (GB) 2015-06-18 WO disclosed