SCHEMBL1679688

SCHEMBL1679688

N[C@@H](CSCNC(=O)O)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ARG1 P05089 1/20 0.48
ARG2 P78540 1/20 0.48
NOS2 P35228 3/20 0.43
NOS1 P29475 2/20 0.43
NOS3 P29474 1/20 0.43
PTGS1 P23219 1/20 0.38
SLC7A11 Q9UPY5 1/20 0.38
KIF11 P52732 3/20 0.38
ALOX15 P16050 2/20 0.37
ALDH1A1 P00352 1/20 0.37
BHMT Q93088 4/20 0.36
SLC7A5 Q01650 1/20 0.35
GRM8 O00222 1/20 0.35
GRM6 O15303 1/20 0.35
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GSR P00390 1/20 0.35
CYP1A2 P05177 1/20 0.35
GRIK1 P39086 1/20 0.35
GRM5 P41594 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1679691 1.00 ARG1 (0.48) ARG1ARG2NOS2NOS1NOS3
SCHEMBL16741952 0.86 ARG1 (0.47) ARG1ARG2NOS2NOS1NOS3
SCHEMBL210388 0.84 NOS2 (0.49) ARG1ARG2NOS2NOS1NOS3
SCHEMBL210387 0.84 NOS2 (0.49) ARG1ARG2NOS2NOS1NOS3
SCHEMBL3928876 0.84 NOS2 (0.49) ARG1ARG2NOS2NOS1NOS3
Hydrochloric Acid SCHEMBL4223453 0.82 NOS2 (0.47) ARG1ARG2NOS2NOS1NOS3
Hydrochloric Acid SCHEMBL29401714 0.82 NOS2 (0.47) ARG1ARG2NOS2NOS1NOS3
Hydrochloric Acid SCHEMBL4223447 0.82 NOS2 (0.47) ARG1ARG2NOS2NOS1NOS3
SCHEMBL11722267 0.81 ARG1 (0.43) ARG1ARG2NOS2NOS1NOS3
SCHEMBL11722274 0.81 ARG1 (0.43) ARG1ARG2NOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10392610-B2 Pregnancy-associated plasma protein-A2 (PAPP-A2) polypeptides COMO BIOTECH APS (DK) 2019-08-27 US disclosed
EP-2339020-B1 Diagnostic methods based on Pregnancy-associated plasma protein-A (PAAP-A) COMO BIOTECH APS (DK) 2017-03-08 EP disclosed
US-20150132770-A1 PREGNANCY-ASSOCIATED PLASMA PROTEIN-A2 (PAPP-A2) POLYNUCLEOTIDES COMO BIOTECH APS (DK) 2015-05-14 US disclosed
US-9005949-B2 Pregnancy-associated plasma protein-A2 (PAPP-A2) polynucleotides COMO BIOTECH APS (DK) 2015-04-14 US disclosed
EP-1346061-B1 PREGNANCY-ASSOCIATED PLASMA PROTEIN-A2 (PAPP-A2) COMO BIOTECH APS (DK) 2014-12-17 EP disclosed
US-20130095569-A1 PREGNANCY-ASSOCIATED PLASMA PROTEIN-A2 (PAPP-A2) POLYNUCLEOTIDES COMO BIOTECH APS (DK) 2013-04-18 US disclosed
US-20130095482-A1 METHODS OF DETECTING PREGNANCY-ASSOCIATED PLASMA PROTEIN-A2 (PAPP-A2) COMO BIOTECH APS (DK) 2013-04-18 US disclosed
EP-2339020-A1 Diagnostic methods based on Pregnancy-associated plasma protein-A (PAAP-A) Como Biotech APS (DK) 2011-06-29 EP disclosed
WO-2011057064-A1 IGF1R INHIBITOR BASED TREATMENT OF PROSTATE CANCER LONG BRIAN (US) 2011-05-12 WO disclosed
US-20110091920-A1 METHOD OF DIAGNOSING A CLINICAL CONDITION BY DETECTION OF A PAPP-A/proMBP COMPLEX COMO BIOTECH APS (DK) 2011-04-21 US disclosed
US-6248869-B1 HUMAN HEART POLYPETIDES; FOR THE DETECTION AND DIAGNOSIS OF HEART INJURY MEDICAL ANALYSIS SYSTEMS, INC. 2001-06-19 US disclosed
WO-2000016704-A1 ULTRASOUND CATHETER FOR IMPROVING BLOOD FLOW TO THE HEART EKOS CORPORATION (US) 2000-03-30 WO disclosed
US-5889147-A OLIGOPEPTIDE, POLYPEPTIDE FROM VENOM OF A CONE SNAIL UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 1999-03-30 US disclosed
WO-1998054218-A1 TROPONIN I FORMS AND USE OF SAME MEDICAL ANALYSIS SYSTEMS INC. (US) 1998-12-03 WO disclosed
WO-1998031705-A1 BROMO-TRYPTOPHAN CONOPEPTIDES UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 1998-07-23 WO disclosed
EP-0805821-A1 HUMAN HEART CNBr TROPONIN I ISOFORM AND USE OF SAME DADE BEHRING INC. (US) 1997-11-12 EP disclosed
WO-1997019955-A1 HUMAN HEART CNBr TROPONIN I ISOFORM AND USE OF SAME DADE INTERNATIONAL INC. (US) 1997-06-05 WO disclosed
US-5464774-A DNA sequence THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1995-11-07 US disclosed
US-5155214-A Basic fibroblast growth factor THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1992-10-13 US disclosed
US-4956455-A POLYPEPTIDES CAPABLE OF STIMULATING GROWTH OF CELLS THE SALK INSTITUTE FOR BIOLOGICAL STUDIES (US) 1990-09-11 US disclosed