SCHEMBL16799581

SCHEMBL16799581

CC1(C)CCCc2nc(OS(=O)(=O)C(F)(F)F)ccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
HTR1D P28221 1/20 0.32
CES2 O00748 2/20 0.31
CES1 P23141 2/20 0.31
DRD1 P21728 1/20 0.31
DRD4 P21917 1/20 0.31
DRD5 P21918 1/20 0.31
HIF1A Q16665 2/20 0.30
EPAS1 Q99814 2/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
APAF1 O14727 1/20 0.30
TERT O14746 1/20 0.30
EED O75530 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
POLB P06746 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14151781 0.77 CNR2 (0.42) DRD2DRD3HTR1DCES1DRD1
SCHEMBL16799475 0.76 DRD2 (0.36) DRD2DRD3CES2CES1DRD1
SCHEMBL1815313 0.72 GRM5 (0.44) KDM4EMEN1ALDH1A1MAPTHPGD
SCHEMBL20365643 0.70 DRD2 (0.34) DRD2DRD3HTR1D
SCHEMBL16799615 0.70 CNR2 (0.33) DRD2DRD3HTR1DDRD4
SCHEMBL8438305 0.70 RXRA (0.40) DRD2DRD3HTR1DDRD4
SCHEMBL20722440 0.69 DRD2 (0.33) DRD2DRD3HTR1D
SCHEMBL30968515 0.69 DRD2 (0.33) DRD2DRD3HTR1D
SCHEMBL20722412 0.69 DRD2 (0.30) DRD2DRD3HTR1D
SCHEMBL30968481 0.69 DRD2 (0.30) DRD2DRD3HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed