SCHEMBL16801258

SCHEMBL16801258

Cc1ccc(-c2ccc3oc4cccc5cccc(c6cccc2c36)c54)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.39
MAOB P27338 7/20 0.39
TNKS O95271 1/20 0.38
PARP1 P09874 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
COMT P21964 1/20 0.37
MAOA P21397 2/20 0.37
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
ENPP1 P22413 2/20 0.36
ENPP3 O14638 1/20 0.36
LMNA P02545 1/20 0.36
RET P07949 1/20 0.36
TSHR P16473 1/20 0.36
ALOX12 P18054 1/20 0.36
KDR P35968 1/20 0.36
HTT P42858 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
AR P10275 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16801277 0.92 ALDH1A1 (0.39) MAOBMAOAALDH1A1ENPP1ENPP3
SCHEMBL16801450 0.90 ALDH1A1 (0.38) MAOBMAOAALDH1A1ENPP1ENPP3
SCHEMBL16801270 0.86 ENPP3 (0.43) MAOBMAOAALDH1A1ENPP1ENPP3
SCHEMBL16801073 0.84 ALDH1A1 (0.40) ADORA3MAOBTNKSPARP1TNKS2
SCHEMBL18159548 0.83 ALDH1A1 (0.38) MAOBMAOAALDH1A1TP53TSHR
SCHEMBL16801129 0.83 ALDH1A1 (0.43) MAOBMAOAALDH1A1TSHRNPC1
SCHEMBL16800612 0.83 ALDH1A1 (0.43) MAOBMAOAALDH1A1TSHRNPC1
SCHEMBL18159552 0.83 HPGD (0.39) MAOAALDH1A1TSHRHTTNPC1
SCHEMBL16801060 0.82 ALDH1A1 (0.36) MAOBMAOAALDH1A1TSHRNPC1
SCHEMBL18159530 0.80 ENPP3 (0.46) MAOBMAOAALDH1A1ENPP1ENPP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015082046-A2 SUBSTITUTED OXEPINES MERCK PATENT GMBH (DE) 2015-06-11 WO disclosed