SCHEMBL16812977

SCHEMBL16812977

O=C1CN=C(c2ccccc2)c2[nH]c3ccccc3c2N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.51
GABRG2 P18507 1/20 0.51
GABRB3 P28472 1/20 0.51
GABRA5 P31644 1/20 0.51
GABRA3 P34903 1/20 0.51
GABRA2 P47869 1/20 0.51
GABRB2 P47870 1/20 0.51
TSHR P16473 2/20 0.47
MAPT P10636 2/20 0.47
ALOX12 P18054 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
PDE4D Q08499 2/20 0.45
CNR1 P21554 1/20 0.45
NTSR1 P30989 1/20 0.45
OPRK1 P41145 1/20 0.45
ALDH1A1 P00352 2/20 0.45
P2RX4 Q99571 2/20 0.44
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
HPGD P15428 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16812974 0.91 SMN1; SMN2 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16812984 0.89 CNR1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16796729 0.87 P2RX4 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16796688 0.87 P2RX4 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16796687 0.87 CYP11B1 (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16813007 0.86 P2RX4 (0.62) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16812980 0.86 ALDH1A1 (0.52) MAPTSMN1; SMN2ALDH1A1HPGDLMNA
SCHEMBL16796606 0.86 P2RX4 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16796615 0.86 P2RX4 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL16812983 0.86 CNR1 (0.47) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed