SCHEMBL16812980

SCHEMBL16812980

COc1ccc(C2=NCC(=O)Nc3c2[nH]c2ccccc32)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 4/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 1/20 0.47
ADORA3 P0DMS8 1/20 0.46
PTGS2 P35354 1/20 0.46
PTGS1 P23219 1/20 0.45
CHRM4 P08173 2/20 0.43
DRD2 P14416 2/20 0.43
HTR7 P34969 2/20 0.43
POLB P06746 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.41
MAPT P10636 2/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16812971 0.87 ALDH1A1 (0.62) ALDH1A1KDM4ESMN1; SMN2HPGDCHRM4
SCHEMBL16812979 0.87 CHRM4 (0.59) ALDH1A1HPGDADORA3CHRM4DRD2
SCHEMBL16812977 0.86 GABRA1 (0.51) ALDH1A1KDM4ESMN1; SMN2LMNAHPGD
SCHEMBL16812984 0.84 CNR1 (0.47) KDM4ESMN1; SMN2LMNAADORA3PTGS2
SCHEMBL16812974 0.83 SMN1; SMN2 (0.44) ALDH1A1SMN1; SMN2MAPTPARP1
SCHEMBL16813010 0.82 ALDH1A1 (0.47) ALDH1A1KDM4ELMNAHPGDCHRM4
SCHEMBL16796608 0.82 ALDH1A1 (0.47) ALDH1A1KDM4EHPGDCHRM4DRD2
SCHEMBL16813047 0.82 PDE9A (0.42) ALDH1A1SMN1; SMN2MAPT
SCHEMBL16812999 0.81 GSK3B (0.44) ALDH1A1LMNAABCG2KMT2ANPC1
SCHEMBL16813001 0.81 SMN1; SMN2 (0.43) SMN1; SMN2ADORA3TNKSPARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed