SCHEMBL1682135

SCHEMBL1682135

NC(=O)c1cc(-c2cccs2)sc1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.61
MAPT P10636 7/20 0.50
ALDH1A1 P00352 7/20 0.50
GAA P10253 6/20 0.50
HPGD P15428 4/20 0.50
KDM4E B2RXH2 3/20 0.50
HSD17B10 Q99714 3/20 0.50
TSHR P16473 1/20 0.50
NPC1 O15118 3/20 0.49
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
MAPK1 P28482 2/20 0.46
PSMD14 O00487 1/20 0.44
MMP2 P08253 1/20 0.44
ALOX15 P16050 1/20 0.44
ADORA1 P30542 1/20 0.43
LMNA P02545 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
GLA P06280 1/20 0.42
CDC7 O00311 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14413993 0.81 MAPT (0.66) MAPTALDH1A1GAAHPGDKDM4E
SCHEMBL4087590 0.77 MAPT (0.68) IKBKBMAPTALDH1A1GAAHPGD
SCHEMBL5898668 0.76 PTK2 (0.54) IKBKBMAPTALDH1A1GAAKDM4E
SCHEMBL3510525 0.76 IKBKB (1.00) IKBKBMAPTALDH1A1GAAHPGD
Carbamic Acid SCHEMBL9378352 0.73 KDM4E (0.52) MAPTALDH1A1GAAHPGDKDM4E
SCHEMBL613585 0.73 IKBKB (0.71) IKBKBMAPTALDH1A1GAAHPGD
SCHEMBL3509823 0.73 IKBKB (0.66) IKBKBMAPTALDH1A1GAAHPGD
SCHEMBL13613456 0.73 CHEK1 (0.57) CDC7CHEK1CHEK2
SCHEMBL3561581 0.72 KCNH2 (0.62) IKBKBHDAC1HDAC3HDAC2
SCHEMBL5898679 0.72 IKBKB (0.64) IKBKBMAPTALDH1A1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046793-A1 NOVEL JAK3 INHIBITOR CONTAINING, AS ACTIVE INGREDIENT, THIOPHENE DERIVATIVE HAVING UREIDO GROUP AND AMINOCARBONYL GROUP AS SUBSTITUENTS 参天製薬株式会社 (JP) 2012-04-12 WO disclosed