SCHEMBL1682282

SCHEMBL1682282

O=S(=O)(c1cccc(F)c1)N(Cc1ccccc1)C1CCN(Cc2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HTR2A P28223 5/20 0.48
HTR2C P28335 1/20 0.48
DRD2 P14416 5/20 0.47
DRD4 P21917 1/20 0.46
HTR1A P08908 3/20 0.46
HTR7 P34969 3/20 0.46
SIGMAR1 Q99720 1/20 0.45
CCR5 P51681 1/20 0.44
RORC P51449 1/20 0.44
OPRM1 P35372 2/20 0.43
CHRM2 P08172 1/20 0.43
CHRM3 P20309 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1682296 0.89 HTR2A (0.53) HTR2AHTR2CDRD2SIGMAR1CCR5
SCHEMBL1682299 0.88 KDM4E (0.49) MEN1KMT2AHTR2AHTR2CDRD2
SCHEMBL1682268 0.88 USP2 (0.55) MEN1KMT2AHTR2ADRD2HTR1A
SCHEMBL1682275 0.87 BCHE (0.49) HTR2AHTR2CDRD2HTR7OPRM1
SCHEMBL1682328 0.83 ALDH1A1 (0.55) KMT2AHTR2AHTR2CHTR1AHTR7
SCHEMBL1682289 0.83 SCN8A (0.49) HTR2AHTR2COPRM1CHRM2CHRM3
SCHEMBL1682312 0.82 HTT (0.54) MEN1KMT2ACHRM2CHRM3ACHE
SCHEMBL1682317 0.82 CHRM4 (0.50) MEN1KMT2AHTR2AHTR2CDRD2
SCHEMBL1682344 0.82 CHRM2 (0.46) OPRM1CHRM2CHRM3
SCHEMBL1682265 0.81 BCHE (0.53) DRD2DRD4SIGMAR1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011043519-A2 SULFONAMIDE DERIVATIVES AS SEROTONIN RECEPTOR ANTAGONIST AND SEROTONIN REUPTAKE INHIBITOR KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2011-04-14 WO claimed
WO-2011043519-A2 SULFONAMIDE DERIVATIVES AS SEROTONIN RECEPTOR ANTAGONIST AND SEROTONIN REUPTAKE INHIBITOR KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2011-04-14 WO disclosed