SCHEMBL168255

SCHEMBL168255

CCS(=O)(=O)c1ccc(C(C)C(=O)OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.44
MMP1 P03956 1/20 0.44
MMP13 P45452 1/20 0.44
PTGS2 P35354 3/20 0.43
RORC P51449 4/20 0.42
GAA P10253 1/20 0.42
MT-CO2 P00403 1/20 0.41
PSIP1 O75475 2/20 0.41
PTGS1 P23219 1/20 0.41
KMT2A Q03164 1/20 0.41
RORA P35398 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12465947 0.87 KMT2A (0.47) HPGDPTGS2RORCGAAPSIP1
SCHEMBL2655181 0.83 AKR1C3 (0.47) HPGDPTGS2MT-CO2PTGS1KMT2A
SCHEMBL166813 0.81 PTGS2 (0.53) PTGS2GAAMT-CO2PSIP1PTGS1
SCHEMBL23174361 0.81 ESR1 (0.45) MMP1MMP13RORCGAAPSIP1
SCHEMBL23174343 0.80 ESR1 (0.44) MMP1MMP13RORCGAAPSIP1
SCHEMBL16879899 0.79 EPHX1 (0.54) RORCGAAPSIP1RORACA12
SCHEMBL17716834 0.78 ALDH1A1 (0.43) HPGDMMP1MMP13RORCGAA
SCHEMBL2601861 0.77 CXCR1 (0.49) HPGDPTGS2PTGS1
SCHEMBL11130803 0.76 HPGD (0.53) HPGDPTGS2MT-CO2PTGS1KMT2A
SCHEMBL12896284 0.76 HPGD (0.53) HPGDPTGS2MT-CO2PTGS1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed
WO-2012028100-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed