SCHEMBL1683428

SCHEMBL1683428

COC(=O)Oc1cn2ncnc(N(C)c3cnc4[nH]ccc4c3)c2c1C(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 12/20 0.51
PDGFRB P09619 2/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
LCK P06239 1/20 0.40
FGFR1 P11362 1/20 0.40
CDK8 P49336 5/20 0.35
KDM5B Q9UGL1 1/20 0.33
PLK4 O00444 1/20 0.32
DCLK1 O15075 1/20 0.32
ROCK2 O75116 1/20 0.32
PRKD3 O94806 1/20 0.32
MAP4K4 O95819 1/20 0.32
PAK4 O96013 1/20 0.32
CHEK2 O96017 1/20 0.32
INSR P06213 1/20 0.32
CDK1 P06493 1/20 0.32
FES P07332 1/20 0.32
ROS1 P08922 1/20 0.32
PDGFRA P16234 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27541332 0.93 KDR (0.51) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683450 0.87 KDR (0.67) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683433 0.81 KDR (0.76) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683443 0.71 KDR (0.61) KDRPDGFRBEGFRERBB2LCK
SCHEMBL5740525 0.68 KDR (0.44) KDREGFRFLT4
SCHEMBL12808319 0.67 KDR (1.00) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683398 0.67 KDR (1.00) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683431 0.67 KDR (1.00) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683459 0.67 KDR (0.84) KDRPDGFRBEGFRERBB2LCK
SCHEMBL1683464 0.67 KDR (0.84) KDRPDGFRBEGFRERBB2LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539763-B1 AZAINDOLE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2011-04-13 EP claimed