SCHEMBL1684264

SCHEMBL1684264

NC(=O)c1cc2n(n1)CCNC2

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.39
CD274 Q9NZQ7 2/20 0.39
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
GSK3B P49841 1/20 0.34
SCN9A Q15858 3/20 0.33
PNMT P11086 1/20 0.33
SOD3 P08294 1/20 0.32
PIM1 P11309 1/20 0.32
PIM3 Q86V86 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
LMNA P02545 1/20 0.31
GRM2 Q14416 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22887771 0.91 CHRNB2 (0.38) PDCD1CD274CHRNB2CHRNA4GSK3B
Hydrochloric Acid SCHEMBL25335409 0.89 CHRNB2 (0.37) PDCD1CD274CHRNB2CHRNA4GSK3B
SCHEMBL30793436 0.89 CHRNB2 (0.35) PDCD1CD274CHRNB2CHRNA4GSK3B
Hydrochloric Acid SCHEMBL25335404 0.88 CHRNB2 (0.36) PDCD1CD274CHRNB2CHRNA4GSK3B
SCHEMBL12282789 0.85 PDCD1 (0.43) PDCD1CD274SOD3HTR2AHTR2C
Hydrochloric Acid SCHEMBL27147176 0.84 PDCD1 (0.42) PDCD1CD274SOD3HTR2AHTR2C
SCHEMBL23652744 0.84 PDCD1 (0.42) PDCD1CD274SCN9APNMTSOD3
SCHEMBL4192949 0.81 PDCD1 (0.38) PDCD1CD274SOD3
SCHEMBL25410303 0.80 BAZ2B (0.43) PDCD1CD274SOD3
SCHEMBL30915369 0.80 PDCD1 (0.40) PDCD1CD274SOD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758585-A4 HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2009-07-22 EP claimed
EP-1758585-A2 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2007-03-07 EP claimed
WO-2005120516-A2 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-12-22 WO claimed
CN-113072551-B Nitrogen-containing biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2024-08-13 CN disclosed
CN-113348170-B Biphenyl derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-22 CN disclosed
WO-2023244713-A1 QUINAZOLINE DERIVATIVES, COMPOSITIONS AND METHODS THEREOF ENSEM THERAPEUTICS, INC. (US) 2023-12-21 WO disclosed
CN-109890819-B Heterocyclic compounds as immunomodulators 因赛特公司 2022-11-22 CN disclosed
EP-4086253-A1 BIPHENYL DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2022-11-09 EP disclosed
WO-2011041512-A2 COMPOSITIONS AND METHODS FOR TREATING MLV-INFECTION, AND PREVENTING AND TREATING MLV-INITIATED DISEASES EMORY UNIVERSITY (US) 2011-04-07 WO disclosed