SCHEMBL16844882

SCHEMBL16844882

COc1ccc(C)c2c1CC(=O)C2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLL Q9UGP5 1/20 0.45
KDM4E B2RXH2 6/20 0.44
ALDH1A1 P00352 5/20 0.44
HPGD P15428 3/20 0.44
GLA P06280 1/20 0.44
GAA P10253 1/20 0.44
ACHE P22303 3/20 0.41
ADRA1A P35348 2/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP19A1 P11511 2/20 0.36
NQO2 P16083 2/20 0.36
MAPT P10636 2/20 0.35
S1PR4 O95977 1/20 0.35
HSP90AA1 P07900 1/20 0.35
G6PD P11413 1/20 0.35
S1PR1 P21453 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6583999 0.89 KDM4E (0.52) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL6272000 0.82 CYP1A2 (0.39) POLLALDH1A1ACHEHSD17B10MAPT
SCHEMBL16835942 0.78 KDM4E (0.43) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL30618055 0.78 KDM4E (0.55) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL8616972 0.78 KDM4E (0.55) KDM4EALDH1A1HPGDGLAGAA
SCHEMBL2722920 0.72 ADRA1A (0.52) POLLKDM4EALDH1A1HPGDGLA
SCHEMBL11985670 0.72 RXRG (0.34) KDM4EALDH1A1HPGDHSD17B10
SCHEMBL1024516 0.71 CES1 (0.36) ALDH1A1HPGDHTR2AHTR2CHTR2B
SCHEMBL2641069 0.71 DRD2 (0.50) ACHEHTR2A
SCHEMBL11985669 0.71 KDM4E (0.41) KDM4EALDH1A1HPGDGLAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015091411-A1 SPIRO-OXAZOLONES F. HOFFMANN-LA ROCHE AG (CH) 2015-06-25 WO disclosed