SCHEMBL16879486

SCHEMBL16879486

N#CCC#CCc1ccc(NC(=O)Cc2ccccn2)nc1F

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
MKNK1 Q9BUB5 1/20 0.38
GLS O94925 12/20 0.38
RAB9A P51151 1/20 0.36
MET P08581 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16879424 0.82 GLS (0.44) CA1CA2CA5ACA7CA5B
SCHEMBL16879101 0.80 DEGS1 (0.47) CA1CA2CA5ACA7CA5B
SCHEMBL16887495 0.78 MKNK1 (0.40) CA1CA2CA5ACA7CA5B
SCHEMBL16879461 0.76 CA1 (0.49) CA1CA2CA5ACA7CA5B
SCHEMBL16879074 0.74 GLS (0.47) GLS
SCHEMBL16887498 0.70 GLS (0.58) GLS
SCHEMBL28803970 0.67 GLS (0.43) CA1CA2CA5ACA7CA5B
SCHEMBL16887488 0.67 MET (0.43) CA1CA2CA5ACA7CA5B
SCHEMBL6622747 0.67 CA1 (0.60) CA1CA2CA5ACA7CA5B
SCHEMBL17223881 0.67 GLS (0.51) CA1CA2CA5ACA7CA5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092235-A2 NOVEL INHIBITORS OF GLUTAMINASE Rhizen Pharmaceuticals S.A. (CH) 2016-11-16 EP disclosed
WO-2015101958-A2 NOVEL INHIBITORS OF GLUTAMINASE RHIZEN PHARMACEUTICALS SA (CH) 2015-07-09 WO disclosed