SCHEMBL16880902

SCHEMBL16880902

COC(=O)c1ccnc(Cc2ccc(CNC(C)=O)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 3/20 0.47
MAP4K1 Q92918 3/20 0.47
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 2/20 0.45
KDM6B O15054 1/20 0.45
KDM5C P41229 1/20 0.45
KDM4C Q9H3R0 1/20 0.45
KDM2A Q9Y2K7 1/20 0.45
KDM3A Q9Y4C1 1/20 0.45
HDAC1 Q13547 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KDM5B Q9UGL1 2/20 0.43
ALDH1A1 P00352 2/20 0.43
RAB9A P51151 2/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
ALOX15 P16050 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
JMJD6 Q6NYC1 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16891458 0.88 KLKB1 (0.49) KLKB1MAP4K1KMT2AKDM5CHDAC1
SCHEMBL16891523 0.84 KDM4E (0.49) KLKB1MAP4K1KDM4EKDM6BKDM5C
SCHEMBL17442609 0.83 KLKB1 (0.66) KLKB1MAP4K1ALOX15
SCHEMBL16880817 0.83 KDM4E (0.48) KLKB1MAP4K1KDM4EKDM6BKDM5C
SCHEMBL581173 0.83 KDM5B (0.56) KMT2AKDM4EKDM6BKDM5CKDM4C
SCHEMBL580585 0.82 KDM5B (0.56) KDM4EKDM6BKDM5CKDM4CKDM2A
SCHEMBL16880900 0.80 KDM4E (0.43) KLKB1MAP4K1KDM4EKDM6BKDM5C
SCHEMBL581445 0.80 MRGPRX4 (0.46) KLKB1MAP4K1KDM4EKDM6BKDM5C
SCHEMBL581463 0.80 PTGS2 (0.46) KLKB1MAP4K1KDM4EKDM6BKDM5C
SCHEMBL581778 0.79 MRGPRX4 (0.56) KMT2AKDM4EKDM6BKDM5CKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3089746-A1 THERAPEUTIC INHIBITORY COMPOUNDS Lifesci Pharmaceuticals, Inc. (BB) 2016-11-09 EP disclosed
WO-2015103317-A1 THERAPEUTIC INHIBITORY COMPOUNDS LIFESCI PHARMACEUTICALS, INC. (BB) 2015-07-09 WO disclosed