SCHEMBL1689094

SCHEMBL1689094

Cc1ccc(-c2ccc(-c3nc4nn(-c5ccccc5)cc4c(=O)n3-c3ccc(Cl)cc3)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
TP53 P04637 2/20 0.48
RAB9A P51151 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MAPT P10636 4/20 0.48
MDM2 Q00987 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
MEN1 O00255 1/20 0.46
HSP90AA1 P07900 1/20 0.46
KMT2A Q03164 1/20 0.46
AURKA O14965 1/20 0.45
CNR1 P21554 2/20 0.45
CNR2 P34972 2/20 0.45
GPR55 Q9Y2T6 2/20 0.45
CCNE1 P24864 2/20 0.43
CDK2 P24941 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PTGS2 P35354 1/20 0.43
GRM5 P41594 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689138 0.99 ALDH1A1 (0.53) ALDH1A1TP53RAB9ANPSR1MAPT
SCHEMBL1689243 0.94 MAPT (0.51) ALDH1A1TP53MAPTGAAMEN1
SCHEMBL5611687 0.92 MAPT (0.52) ALDH1A1MAPTMDM2GAAMEN1
SCHEMBL1689133 0.91 MAPT (0.58) ALDH1A1TP53RAB9ANPSR1MAPT
SCHEMBL5612533 0.90 MAPT (0.45) ALDH1A1NPSR1MAPTMEN1HSP90AA1
SCHEMBL1688969 0.89 MAPT (0.49) ALDH1A1MAPTMEN1HSP90AA1KMT2A
SCHEMBL5611548 0.89 TP53 (0.61) ALDH1A1TP53RAB9ANPSR1MAPT
SCHEMBL5611531 0.89 TP53 (0.46) ALDH1A1TP53MAPTMDM2LMNA
SCHEMBL1689182 0.89 MAPT (0.43) ALDH1A1TP53RAB9ANPSR1MAPT
SCHEMBL1688924 0.89 MAPT (0.43) ALDH1A1TP53MAPTMEN1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807429-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM, LLC (BM) 2007-07-18 EP claimed
WO-2006047516-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2006-05-04 WO claimed