SCHEMBL16900147

SCHEMBL16900147

CC(C)(C)OC(=O)CN1CCC(N)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
WNT1 P04628 1/20 0.38
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
HTR4 Q13639 1/20 0.38
PLA2G10 O15496 2/20 0.38
PLA2G5 P39877 2/20 0.38
CNR1 P21554 1/20 0.36
GNAI3 P08754 2/20 0.35
GNAO1 P09471 2/20 0.35
GNAI1 P63096 2/20 0.35
CDK9 P50750 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
HPGD P15428 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL572705 0.84 CHRM2 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL13698802 0.84 SMN1; SMN2 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL6217337 0.83 HTR4 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL8486056 0.83 SMN1; SMN2 (0.54) WNT1GSK3BDYRK1ASMN1; SMN2CHRM1
SCHEMBL3470166 0.83 PLA2G10 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL3799622 0.83 PLA2G10 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL27147241 0.83 PLA2G10 (0.41) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL14436566 0.83 HSD11B1 (0.40) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL25355009 0.82 PLA2G10 (0.40) WNT1GSK3BDYRK1AHTR4PLA2G10
SCHEMBL18173283 0.81 NR1H2 (0.43) WNT1GSK3BDYRK1AHTR4PLA2G10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861577-B1 TERTIARY AMINES, MEDICAMENTS CONTAINING SAID AMINES, USE THEREOF AND PROCESSES FOR THE PREPARATION THEREOF BOEHRINGER INGELHEIM INT (DE) 2017-01-04 EP disclosed
US-9078909-B2 Tertiary amines, medicaments containing said amines, use thereof and processes for the preparation thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-07-14 US disclosed
US-9078909-B2 Tertiary amines, medicaments containing said amines, use thereof and processes for the preparation thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-07-14 US disclosed