SCHEMBL16900352

SCHEMBL16900352

Cc1ccc2c(c1)c1c(n2CCc2ccc(CF)nc2)CN2CCC1C2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 15/20 0.48
HTR6 P50406 13/20 0.48
ADRA2A P08913 3/20 0.48
HTR2A P28223 3/20 0.48
HTR2C P28335 3/20 0.48
HTR7 P34969 3/20 0.48
ADRA1A P35348 3/20 0.48
DRD2 P14416 2/20 0.48
BCHE P06276 1/20 0.48
ADRA2B P18089 1/20 0.48
ADRA2C P18825 1/20 0.48
ACHE P22303 1/20 0.48
HRH2 P25021 1/20 0.48
ADRA1D P25100 1/20 0.48
HTR1D P28221 1/20 0.48
HTR1E P28566 1/20 0.48
ADRA1B P35368 1/20 0.48
DRD3 P35462 1/20 0.48
HTR2B P41595 1/20 0.48
HTR5A P47898 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12243933 0.90 HRH1 (0.61) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL12243902 0.87 HRH1 (0.47) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL12243987 0.82 HRH1 (0.59) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL12243922 0.82 HRH1 (0.45) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL12243928 0.80 HTR6 (0.61) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL15868830 0.77 HRH1 (0.66) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL16638515 0.77 HTR6 (0.44) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL18155238 0.77 HRH1 (0.67) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL15868829 0.77 HTR6 (0.80) HRH1HTR6ADRA2AHTR2AHTR2C
SCHEMBL1445544 0.76 HDAC2 (0.43) HRH1HTR6ADRA2AHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9271971-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2016-03-01 US disclosed
US-9085580-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2015-07-21 US disclosed
US-9079904-B2 Pyrido[3,4-B]indoles and methods of use MEDIVATION TECHNOLOGIES, INC. (US) 2015-07-14 US disclosed