SCHEMBL16907488

SCHEMBL16907488

COc1ccc(CSc2ccc(N)c3nonc23)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 4/20 0.42
GSTM2 P28161 4/20 0.42
TSHR P16473 2/20 0.42
APP P05067 1/20 0.41
IDO1 P14902 2/20 0.40
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KMT2A Q03164 2/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16907678 0.85 GSTP1 (0.48) GSTP1GSTM2TSHRAPPIDO1
SCHEMBL16907548 0.81 CA1 (0.47) GSTP1GSTM2TSHRAPPSMN1; SMN2
SCHEMBL22705031 0.80 CYP1A2 (0.40) TSHRAPPIDO1LMNAMAPT
SCHEMBL298137 0.79 GSTP1 (0.72) GSTP1GSTM2IDO1
SCHEMBL7298052 0.73 POLB (0.65) TSHRAPPIDO1LMNAMAPT
SCHEMBL22689283 0.71 ALDH1A1 (0.45) LMNAMAPTL3MBTL1KMT2AHPGD
SCHEMBL22704877 0.71 SMN1; SMN2 (0.36) IDO1LMNAMAPTHPGDCYP1A2
SCHEMBL7291905 0.70 CYP1A2 (0.45) TSHRAPPIDO1KMT2AMAOA
SCHEMBL13457191 0.70 CYP1A2 (0.45) TSHRAPPIDO1LMNAMAPT
SCHEMBL10687383 0.70 APP (0.58) TSHRAPPIDO1LMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020234424-A1 BENZO[C][1,2,5]OXADIAZOLE FOR THE TREATMENT OF DISEASES CAUSED BY HELICOBACTER UNIVERSIDAD DE ZARAGOZA (ES) 2020-11-26 WO disclosed
WO-2015104433-A1 BENZO[C][1,2,5]OXADIAZOLE DERIVATIVES FOR TREATING DISEASES CAUSED BY HELICOBACTER UNIVERSIDAD DE ZARAGOZA (ES) 2015-07-16 WO disclosed