SCHEMBL16927161

SCHEMBL16927161

O=C1c2ccc(C#Cc3ccccc3)cc2C(=O)N1c1ccc(N2C(=O)c3ccc(C#Cc4ccccc4)cc3C2=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.54
ESR1 P03372 3/20 0.54
ESR2 Q92731 2/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
SCN2A Q99250 1/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
GFER P55789 1/20 0.47
NPC1 O15118 1/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.45
CASP1 P29466 1/20 0.45
RAB9A P51151 1/20 0.45
CASP7 P55210 1/20 0.45
HSD17B10 Q99714 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678431 0.97 ESR1 (0.58) GRM5ESR1ESR2CA12CA1
SCHEMBL20716046 0.94 ALDH1A1 (0.55) GRM5ESR1CA12CA1CA2
SCHEMBL2471106 0.93 ESR1 (0.63) GRM5ESR1ESR2CA12CA1
SCHEMBL2625350 0.93 GRM5 (0.48) GRM5ESR1ESR2CA12CA1
SCHEMBL13433471 0.90 GRM5 (0.51) GRM5ESR1SCN2AMEN1KMT2A
SCHEMBL16937189 0.90 GRM5 (0.51) GRM5ESR1SCN2AMEN1KMT2A
SCHEMBL13900300 0.90 CA9 (0.66) ESR1CA12CA1CA2CA9
SCHEMBL29637688 0.90 CA9 (0.66) ESR1CA12CA1CA2CA9
SCHEMBL28947748 0.90 ESR1 (0.51) GRM5ESR1ESR2CA12CA1
SCHEMBL13900322 0.89 CA9 (0.55) GRM5ESR1ESR2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2899179-A1 Combination of cross-linkers including carbon-carbon triple bonds Nexam Chemical AB (SE) 2015-07-29 EP disclosed