SCHEMBL169435

SCHEMBL169435

COCNc1ccc(C2CCN(C(=O)OCc3ccccc3)CC2)nc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 10/20 0.53
CYP2D6 P10635 4/20 0.53
CYP2C9 P11712 4/20 0.53
CYP3A4 P08684 3/20 0.53
SMN1; SMN2 Q16637 3/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
HTT P42858 1/20 0.49
CYP2C19 P33261 1/20 0.48
TRPC3 Q13507 2/20 0.47
TRPC7 Q9HCX4 2/20 0.47
JAK2 O60674 2/20 0.47
JAK1 P23458 2/20 0.47
TYK2 P29597 2/20 0.47
JAK3 P52333 2/20 0.47
ENPP2 Q13822 1/20 0.46
DGAT1 O75907 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171606 0.90 JAK2 (0.49) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL14544121 0.88 GRIN2B (0.52) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL171472 0.83 SMN1; SMN2 (0.58) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL169370 0.80 SMN1; SMN2 (0.57) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL171583 0.80 SMN1; SMN2 (0.57) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL171605 0.80 SMN1; SMN2 (0.58) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL13490558 0.79 SMN1; SMN2 (0.59) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL171543 0.78 GRIN2B (0.42) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2
SCHEMBL171368 0.78 NAMPT (0.49) GRIN2BCYP2D6CYP2C9CYP3A4
SCHEMBL171621 0.78 GRIN2B (0.53) GRIN2BCYP2D6CYP2C9CYP3A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426120-A1 Pyridyltetrahydropyridines and pyridylpiperidines, and method of manufacturing them Fujifilm Finechemicals Co., Ltd. (JP) 2012-03-07 EP disclosed