SCHEMBL171606

SCHEMBL171606

COCNc1ccc(C2CCCN(C(=O)OCc3ccccc3)C2)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 3/20 0.49
JAK1 P23458 3/20 0.49
TYK2 P29597 2/20 0.49
JAK3 P52333 2/20 0.49
GRIN2B Q13224 6/20 0.46
CYP2D6 P10635 4/20 0.46
CYP2C9 P11712 4/20 0.46
CYP3A4 P08684 3/20 0.46
MAPK1 P28482 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PDE4B Q07343 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
BCL9 O00512 1/20 0.43
CTNNB1 P35222 1/20 0.43
LCK P06239 2/20 0.43
USP30 Q70CQ3 1/20 0.43
HTT P42858 1/20 0.43
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169435 0.90 GRIN2B (0.53) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL14544157 0.89 JAK2 (0.50) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490610 0.83 BCL9 (0.52) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490733 0.81 RET (0.44) JAK2JAK1TYK2JAK3CYP2D6
SCHEMBL169477 0.80 JAK2 (0.49) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL171665 0.80 JAK2 (0.52) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490730 0.80 JAK2 (0.50) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490607 0.79 JAK2 (0.48) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490606 0.79 JAK2 (0.46) JAK2JAK1TYK2JAK3GRIN2B
SCHEMBL13490506 0.79 JAK2 (0.55) JAK2JAK1TYK2JAK3GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426120-A1 Pyridyltetrahydropyridines and pyridylpiperidines, and method of manufacturing them Fujifilm Finechemicals Co., Ltd. (JP) 2012-03-07 EP disclosed
US-7632950-B2 Pyridyltetrahydropyridines and pyridylpiperidines and method of manufacturing them FUJIFILM FINECHEMICALS CO., LTD (JP) 2009-12-15 US disclosed