SCHEMBL169475

SCHEMBL169475

NC(=O)[C@@H](N)CC[C]=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5557115 1.00
SCHEMBL61372 1.00
SCHEMBL157042 0.80
SCHEMBL639292 0.80
SCHEMBL157041 0.80
SCHEMBL14956926 0.78 ALOX15 (0.43)
SCHEMBL17541311 0.78 ALOX15 (0.43)
SCHEMBL15676365 0.78 ALOX15 (0.43)
SCHEMBL20924801 0.74 ALOX15 (0.37)
SCHEMBL7398604 0.74

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 168 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20030147898-A1 Adjuvant formulation comprising a submicron oil droplet emulson NOVARTIS VACCINES AND DIAGNOSTICS, INC. 2003-08-07 US claimed
EP-0489153-B1 VACCINE COMPOSITIONS CONTAINING LIPOSOMES CHIRON CORP (US) 1999-10-13 EP claimed
WO-1998009989-A1 THE USE OF MURAMYLPEPTIDES IN THE TREATMENT OF MYELOSUPPRESSED OR OTHERWISE IMMUNOCOMPROMISED STATES PEPTECH (UK) LIMITED (GB) 1998-03-12 WO claimed
US-5709879-A Vaccine compositions containing liposomes CHIRON CORPORATION (US) 1998-01-20 US claimed
EP-0782454-A1 USE OF MURAMYL PEPTIDE COMPOUNDS PEPTECH (UK) (GB) 1997-07-09 EP claimed
EP-0768888-A1 USE OF MURAMYL PEPTIDE COMPOUNDS PEPTECH (UK) LIMITED (GB) 1997-04-23 EP claimed
EP-0722332-A1 COMPOUNDS FOR MEDICINAL USE PEPTECH (UK) LIMITED (GB) 1996-07-24 EP claimed
WO-1996009063-A1 USE OF MURAMYL PEPTIDE COMPOUNDS PEPTECH(UK) LIMITED (GB) 1996-03-28 WO claimed
WO-1996001645-A1 USE OF MURAMYL PEPTIDE COMPOUNDS PEPTECH(UK) LIMITED (GB) 1996-01-25 WO claimed
WO-1995010293-A1 COMPOUNDS FOR MEDICINAL USE PEPTECH (UK) LIMITED (GB) 1995-04-20 WO claimed
EP-0627928-A1 USE OF MURAMYL PEPTIDE FOR THE TREATMENT OF TOXICITY PEPTECH (UK) (GB) 1994-12-14 EP claimed
EP-0399843-B1 Adjuvant formulation comprising a submicron oil droplet emulsion CHIRON CORP (US) 1994-07-13 EP claimed
EP-0489153-A4 VACCINE COMPOSITIONS CONTAINING LIPOSOMES 1993-04-21 EP claimed
EP-0280610-B1 DIPEPTIDES, PREPARATION PROCESS AND USE IN DOSING PROTEASES SERBIO (FR) 1992-10-21 EP claimed
EP-0489153-A1 VACCINE COMPOSITIONS CONTAINING LIPOSOMES CHIRON CORPORATION (US) 1992-06-10 EP claimed
WO-1992000081-A1 VACCINE COMPOSITIONS CONTAINING LIPOSOMES CHIRON CORPORATION (US) 1992-01-09 WO claimed
WO-1990014837-A1 ADJUVANT FORMULATION COMPRISING A SUBMICRON OIL DROPLET EMULSION CHIRON CORPORATION (US) 1990-12-13 WO claimed
EP-0213523-B1 PHARMACEUTICAL COMPOSITIONS CONTAINING ACYLATED PHOSPHOLIPIDS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1990-12-12 EP claimed
EP-0399843-A2 Adjuvant formulation comprising a submicron oil droplet emulsion CHIRON CORPORATION (US) 1990-11-28 EP claimed
EP-0178624-B1 LIPOSOMES FROM SYNTHETIC LIPIDS CIBA-GEIGY AG (CH) 1990-11-22 EP claimed