SCHEMBL1695601

SCHEMBL1695601

CO/C(=C\c1ccccc1)C(=O)NN

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 6/20 0.56
AKR1C3 P42330 1/20 0.44
LMNA P02545 2/20 0.43
KMT2A Q03164 5/20 0.43
MEN1 O00255 4/20 0.43
MAPT P10636 2/20 0.43
RECQL P46063 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 1/20 0.41
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
NFKB1 P19838 1/20 0.41
RAB9A P51151 1/20 0.41
NFKB2 Q00653 1/20 0.41
RELA Q04206 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1695603 1.00 ABCG2 (0.56) ABCG2AKR1C3LMNAKMT2AMEN1
SCHEMBL11026391 0.86 ABCG2 (0.56) ABCG2AKR1C3LMNAKMT2AMEN1
SCHEMBL25728780 0.84 ABCG2 (0.57) ABCG2AKR1C3LMNAKMT2AMEN1
SCHEMBL7672337 0.81 ABCG2 (0.51) ABCG2AKR1C3KMT2AMEN1RECQL
SCHEMBL5698609 0.81 MEN1 (0.42) ABCG2AKR1C3LMNAKMT2AMEN1
SCHEMBL83065 0.81 AKR1C3 (0.55) ABCG2AKR1C3KMT2AMEN1RECQL
SCHEMBL3818255 0.81 AKR1C3 (0.55) ABCG2AKR1C3KMT2AMEN1RECQL
SCHEMBL9103420 0.81 ABCG2 (0.54) ABCG2AKR1C3KMT2AMEN1MAPT
SCHEMBL3485765 0.81 AKR1C3 (0.55) ABCG2AKR1C3KMT2AMEN1RECQL
SCHEMBL31439245 0.81 MAPT (0.60) ABCG2LMNAKMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138657-A1 ARYL SUBSTITUTED OLEFINIC COMPOUNDS AS PDE10A INHIBITORS GLENMARK PHARMACEUTICALS S.A. (CH) 2011-11-10 WO disclosed