SCHEMBL16964802

SCHEMBL16964802

O=C1CCC(=O)N1CC1CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.43
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
POLB P06746 2/20 0.36
CYP1B1 Q16678 1/20 0.35
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
KMT2A Q03164 1/20 0.33
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23476568 0.89 HTR1A (0.38) HTR1APSEN1PSEN2APH1BNCSTN
SCHEMBL19091274 0.88 CHRM5 (0.43) HTR1ACYP1B1CHRM2CHRM4CHRM5
SCHEMBL1920814 0.85 HTR1A (0.37) HTR1APSEN1PSEN2APH1BNCSTN
SCHEMBL2519541 0.85 HTR1A (0.37) HTR1APSEN1PSEN2APH1BNCSTN
SCHEMBL535579 0.84 PLG (0.47) HTR1APOLBSMN1; SMN2MEN1ALDH1A1
SCHEMBL16552327 0.84 PLG (0.47) HTR1APOLBSMN1; SMN2MEN1ALDH1A1
SCHEMBL17532449 0.83 HTR1A (0.37) HTR1APSEN1PSEN2APH1BNCSTN
SCHEMBL17145362 0.82 SMN1; SMN2 (0.38) HTR1APOLBSMN1; SMN2MEN1ALDH1A1
SCHEMBL23476597 0.82 SMN1; SMN2 (0.38) HTR1APOLBSMN1; SMN2MEN1ALDH1A1
SCHEMBL10082604 0.82 HTT (0.37) HTR1APOLBSMN1; SMN2RAB9AADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900242-A1 SUBSTITUTED CYCLOPROPYL COMPOUNDS Merck Sharp & Dohme Corp. (US) 2015-08-05 EP disclosed