SCHEMBL16965645

SCHEMBL16965645

CCc1nc2cc(C)c(C)nc2n1Cc1ccc(C=CCN2CCN(CCN3CCOCC3)CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GPR4 P46093 10/20 0.55
KCNH2 Q12809 3/20 0.55
HRH3 Q9Y5N1 3/20 0.55
TRPC5 Q9UL62 1/20 0.38
BRD4 O60885 8/20 0.37
CREBBP Q92793 8/20 0.37
PDE10A Q9Y233 1/20 0.37
EP300 Q09472 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16965545 0.91 GPR4 (0.58) GPR4KCNH2HRH3
SCHEMBL16964963 0.88 GPR4 (0.59) GPR4KCNH2HRH3
SCHEMBL16965643 0.86 GPR4 (0.73) GPR4KCNH2HRH3
SCHEMBL16964742 0.86 GPR4 (0.55) GPR4KCNH2HRH3
SCHEMBL13578526 0.85 GPR4 (0.76) GPR4KCNH2HRH3
SCHEMBL16968375 0.85 GPR4 (0.76) GPR4KCNH2HRH3
Hydrochloric Acid SCHEMBL4326596 0.84 GPR4 (0.75) GPR4KCNH2HRH3
Hydrochloric Acid SCHEMBL4326590 0.84 GPR4 (0.75) GPR4KCNH2HRH3
SCHEMBL16964531 0.83 GPR4 (0.61) GPR4KCNH2HRH3
SCHEMBL16964709 0.82 GPR4 (0.50) GPR4KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900237-A1 COMPOUNDS FOR USE IN GASTRIC COMPLICATION Novartis AG (CH) 2015-08-05 EP disclosed