SCHEMBL16965643

SCHEMBL16965643

CCc1nc2cc(C)c(C)nc2n1Cc1ccc(C=CCN2CCN(C(C)C)CC2)cc1

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR4 P46093 18/20 0.73
KCNH2 Q12809 3/20 0.73
HRH3 Q9Y5N1 3/20 0.73
ALDH1A1 P00352 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16964531 0.91 GPR4 (0.61) GPR4KCNH2HRH3
SCHEMBL16965545 0.90 GPR4 (0.58) GPR4KCNH2HRH3ALDH1A1
SCHEMBL16965452 0.90 GPR4 (0.72) GPR4KCNH2HRH3ALDH1A1PKM
SCHEMBL16964963 0.89 GPR4 (0.59) GPR4KCNH2HRH3
SCHEMBL16964742 0.87 GPR4 (0.55) GPR4KCNH2HRH3
SCHEMBL16965645 0.86 GPR4 (0.55) GPR4KCNH2HRH3
SCHEMBL16965751 0.85 GPR4 (0.59) GPR4KCNH2HRH3ALDH1A1PKM
SCHEMBL4326230 0.84 GPR4 (1.00) GPR4KCNH2HRH3
SCHEMBL4326234 0.84 GPR4 (1.00) GPR4KCNH2HRH3
SCHEMBL16964709 0.81 GPR4 (0.50) GPR4KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900237-A1 COMPOUNDS FOR USE IN GASTRIC COMPLICATION Novartis AG (CH) 2015-08-05 EP claimed
EP-2900237-A1 COMPOUNDS FOR USE IN GASTRIC COMPLICATION Novartis AG (CH) 2015-08-05 EP disclosed