SCHEMBL16965751

SCHEMBL16965751

Cc1cc2nc(C(F)(F)F)n(Cc3ccc(C=CCN4CCN(C(C)C)CC4)cc3)c2nc1C

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR4 P46093 13/20 0.59
KCNH2 Q12809 4/20 0.56
HRH3 Q9Y5N1 3/20 0.56
PKM P14618 2/20 0.35
ALDH1A1 P00352 2/20 0.34
GAA P10253 2/20 0.34
CYP3A4 P08684 3/20 0.33
HIF1A Q16665 3/20 0.33
LMNA P02545 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
MAPK1 P28482 2/20 0.33
GMNN O75496 1/20 0.33
ABCB11 O95342 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM4 P08173 1/20 0.33
HTR1A P08908 1/20 0.33
CHRM5 P08912 1/20 0.33
ADRA2A P08913 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16965452 0.88 GPR4 (0.72) GPR4KCNH2HRH3PKMALDH1A1
SCHEMBL16965643 0.85 GPR4 (0.73) GPR4KCNH2HRH3PKMALDH1A1
SCHEMBL4369299 0.85 GPR4 (0.79) GPR4KCNH2HRH3
SCHEMBL4369304 0.85 GPR4 (0.79) GPR4KCNH2HRH3
Hydrochloric Acid SCHEMBL4368771 0.84 GPR4 (0.77) GPR4KCNH2HRH3
Hydrochloric Acid SCHEMBL4368767 0.84 GPR4 (0.77) GPR4KCNH2HRH3
Hydrochloric Acid SCHEMBL4470674 0.81 GPR4 (0.41) GPR4KCNH2HRH3ALDH1A1LMNA
SCHEMBL16964531 0.77 GPR4 (0.61) GPR4KCNH2HRH3
SCHEMBL16964963 0.75 GPR4 (0.59) GPR4KCNH2HRH3MAPK1
SCHEMBL16965545 0.75 GPR4 (0.58) GPR4KCNH2HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900237-A1 COMPOUNDS FOR USE IN GASTRIC COMPLICATION Novartis AG (CH) 2015-08-05 EP disclosed