SCHEMBL16972717

SCHEMBL16972717

CCc1c(-c2ccc(N3CC[C@@H](O)C3)cc2)[nH]c(=O)c2c(=O)[nH]sc12

nearest known ligand 0.76

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.76
WDR91 A4D1P6 1/20 0.35
SYK P43405 5/20 0.34
PRKAG1 P54619 1/20 0.34
PRKAA1 Q13131 1/20 0.34
PRKAB1 Q9Y478 1/20 0.34
MAPT P10636 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16984241 1.00 KCNH2 (0.76) KCNH2WDR91SYKPRKAG1PRKAA1
SCHEMBL16972707 0.86 KCNH2 (0.73) KCNH2
SCHEMBL16984195 0.86 KCNH2 (0.73) KCNH2
SCHEMBL16972703 0.86 KCNH2 (1.00) KCNH2SYK
SCHEMBL16984191 0.85 KCNH2 (0.72) KCNH2
SCHEMBL16972673 0.81 KCNH2 (0.66) KCNH2
SCHEMBL16972700 0.80 KCNH2 (0.64) KCNH2
SCHEMBL16972732 0.79 KCNH2 (0.64) KCNH2
SCHEMBL16972693 0.79 KCNH2 (0.61) KCNH2
SCHEMBL16972695 0.79 KCNH2 (0.61) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed