SCHEMBL16972732

SCHEMBL16972732

CCc1c(-c2ccc(N3CC4CCCN(C)C4C3)cc2)[nH]c(=O)c2c(=O)[nH]sc12

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.64
HRH3 Q9Y5N1 3/20 0.39
CHRNA7 P36544 1/20 0.33
KMT5A Q9NQR1 1/20 0.31
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972673 0.95 KCNH2 (0.66) KCNH2HRH3CHRNA7
SCHEMBL16984241 0.79 KCNH2 (0.76) KCNH2
SCHEMBL16972717 0.79 KCNH2 (0.76) KCNH2
SCHEMBL16984195 0.78 KCNH2 (0.73) KCNH2HRH3
SCHEMBL16972703 0.78 KCNH2 (1.00) KCNH2
SCHEMBL16972707 0.78 KCNH2 (0.73) KCNH2HRH3
SCHEMBL16984191 0.77 KCNH2 (0.72) KCNH2
SCHEMBL16972700 0.75 KCNH2 (0.64) KCNH2
SCHEMBL16972693 0.73 KCNH2 (0.61) KCNH2
SCHEMBL16972695 0.73 KCNH2 (0.61) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed