SCHEMBL16975058

SCHEMBL16975058

CCCCCCc1sc2nc[nH]c(=O)c2c1Br

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.44
PDPK1 O15530 1/20 0.44
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
LMNA P02545 1/20 0.41
BCAT2 O15382 1/20 0.40
CYP1A2 P05177 1/20 0.39
TMIGD3 P0DMS9 1/20 0.39
CYP2C9 P11712 1/20 0.39
ADORA1 P30542 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
CHEK1 O14757 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16975093 0.89 PDPK1 (0.49) HTTPDPK1KDM4EGAALMNA
SCHEMBL3100667 0.85 PDPK1 (0.56) HTTPDPK1KDM4EGAALMNA
SCHEMBL3102508 0.84 PDPK1 (0.57) HTTPDPK1KDM4EGAALMNA
SCHEMBL16975043 0.83 PDPK1 (0.51) HTTPDPK1KDM4EGAALMNA
SCHEMBL3102176 0.80 PDPK1 (0.59) HTTPDPK1KDM4EGAALMNA
SCHEMBL3114173 0.77 PDPK1 (0.59) HTTPDPK1KDM4EGAALMNA
SCHEMBL3103014 0.76 PDPK1 (0.50) HTTPDPK1KDM4EGAALMNA
SCHEMBL16982857 0.72 PDPK1 (0.70) HTTPDPK1KDM4EGAALMNA
SCHEMBL7919295 0.72 PDPK1 (0.54) HTTPDPK1KDM4EGAALMNA
SCHEMBL3095187 0.70 TMIGD3 (0.69) HTTPDPK1KDM4EGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114663-A1 NOVEL THIENO [2,3-D]PYRIMIDIN-4(3H)-ONE COMPOUNDS WITH ANTIMYCOBACTERIAL PROPERTIES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-08-06 WO claimed