SCHEMBL169816

SCHEMBL169816

COC(=O)c1[nH]nc(C)c1I

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.50
ALDH1A1 P00352 5/20 0.40
HSD17B10 Q99714 4/20 0.40
GAA P10253 1/20 0.39
AR P10275 1/20 0.39
MAPK1 P28482 1/20 0.38
PDE4D Q08499 1/20 0.38
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
NPSR1 Q6W5P4 2/20 0.35
POLB P06746 2/20 0.35
RAB9A P51151 2/20 0.35
ALPL P05186 2/20 0.35
CSNK2A2 P19784 1/20 0.35
KDR P35968 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
KDM4E B2RXH2 1/20 0.34
STAT3 P40763 1/20 0.34
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18560457 0.81 KDM4C (0.65) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL7902863 0.80 KDM4C (0.53) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL23115860 0.78 KDM4C (0.67) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL23294471 0.77 KDM4C (0.50) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL11204987 0.74 KDM4C (0.47) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL171417 0.73 KDM4C (0.46) KDM4CALDH1A1HSD17B10GAAAR
SCHEMBL30975958 0.72 ALDH1A1 (0.44) KDM4CALDH1A1HSD17B10MAPK1LMNA
SCHEMBL30976062 0.72 KDM4C (0.41) KDM4CALDH1A1HSD17B10MAPK1LMNA
SCHEMBL30976137 0.71 KDM4C (0.41) KDM4CALDH1A1HSD17B10MAPK1LMNA
SCHEMBL30975871 0.71 KDM4C (0.41) KDM4CALDH1A1HSD17B10MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118930533-A Substituted pyrazole compounds and methods of using the same for treating hyperproliferative diseases 班塔姆制药有限责任公司 2024-11-12 CN disclosed
CN-110603254-B Substituted pyrazole compounds and methods of using the same for treating hyperproliferative diseases 班塔姆制药有限责任公司 2024-04-12 CN disclosed
EP-2426110-A1 PYRAZOLYL ACRYLONITRILE COMPOUNDS AND USES THEREOF Sinochem Corporation (CN) 2012-03-07 EP disclosed