SCHEMBL7902863

SCHEMBL7902863

COC(=O)c1[nH]nc(C)c1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.53
ALDH1A1 P00352 5/20 0.41
HSD17B10 Q99714 3/20 0.41
AR P10275 1/20 0.41
MAPK1 P28482 1/20 0.40
PDE4D Q08499 1/20 0.40
DYRK1A Q13627 1/20 0.39
NPSR1 Q6W5P4 2/20 0.39
LMNA P02545 3/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 1/20 0.37
TSHR P16473 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CSNK2A2 P19784 1/20 0.37
KDR P35968 1/20 0.37
CSNK2B P67870 1/20 0.37
CSNK2A1 P68400 1/20 0.37
ALPL P05186 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23115860 0.82 KDM4C (0.67) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL169816 0.80 KDM4C (0.50) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL27140315 0.80 PDE4D (0.59) ALDH1A1HSD17B10MAPK1PDE4DLMNA
SCHEMBL9038005 0.80 KDM4C (0.50) KDM4CALDH1A1HSD17B10MAPK1NPSR1
SCHEMBL23294471 0.80 KDM4C (0.50) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL4650087 0.80 KDM4C (0.50) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL11204987 0.77 KDM4C (0.47) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL11205400 0.77 KDM4C (0.47) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL171417 0.76 KDM4C (0.46) KDM4CALDH1A1HSD17B10ARMAPK1
SCHEMBL20471480 0.76 KDM4C (0.46) KDM4CALDH1A1HSD17B10MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112824393-A Preparation method of 3, 4-dimethylpyrazole-5-formate compound 中国科学院大连化学物理研究所 2021-05-21 CN disclosed
CN-106608873-A Pyrazole amide compound, and preparation method and application thereof 湖南化工研究院有限公司 2017-05-03 CN disclosed
US-6297386-B1 BY REACTING THE ENOLATE OF A 2,4-DIKETOCARBOXYLIC ESTER IN THE PRESENCE OF A SOLVENT AND WATER WITH AN N-ALKYLHYDRAZINIUM SALT,PARTICULARLY ECONOMICAL PREPARATION OF AND WITH ONLY LIMITED FORMATION OF UNDESIRABLE ISOMERS. PATENT NUMBER: BAYER AKTIENGESELLSCHAFT (DE) 2001-10-02 US disclosed
US-5977378-A Process for the preparation of 1-alkyl-pyrazole-5-carboxylic acid esters BAYER AKTIENGESELLSCHAFT (DE) 1999-11-02 US disclosed