SCHEMBL1698717

SCHEMBL1698717

CC(C)(F)c1cc(NC(=O)Nc2ccc(NC(=O)c3ccc(OC4CC(C)(C)[N+](C)(OS(C)(=O)=O)C(C)(C)C4)cn3)cc2)on1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 11/20 0.52
CSF1R P07333 10/20 0.52
PDGFRB P09619 3/20 0.52
KIT P10721 3/20 0.52
PDGFRA P16234 3/20 0.52
MAPK14 Q16539 3/20 0.40
RAF1 P04049 2/20 0.40
BRAF P15056 2/20 0.38
EPHX2 P34913 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1698965 0.95 FLT3 (0.55) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698712 0.86 FLT3 (0.68) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL15388274 0.86 FLT3 (0.54) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698946 0.86 FLT3 (0.62) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698798 0.85 FLT3 (0.73) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698846 0.84 FLT3 (0.72) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698736 0.84 FLT3 (0.63) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698861 0.83 FLT3 (0.51) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698962 0.81 FLT3 (0.71) FLT3CSF1RPDGFRBKITPDGFRA
SCHEMBL1698857 0.79 CSF1R (0.68) FLT3CSF1RPDGFRBKITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130310357-A1 Azolyl Urea Compounds and Methods of Use Thereof AMBIT BIOSCIENCES CORPORATION (US) 2013-11-21 US claimed
WO-2011150198-A1 AZOLYL UREA COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2011-12-01 WO claimed
US-9296722-B2 Azolyl urea compounds and methods of use thereof AMBIT BIOSCIENCES CORPORATION (US) 2016-03-29 US disclosed
US-20130310357-A1 Azolyl Urea Compounds and Methods of Use Thereof AMBIT BIOSCIENCES CORPORATION (US) 2013-11-21 US disclosed
WO-2011150198-A1 AZOLYL UREA COMPOUNDS AND METHODS OF USE THEREOF AMBIT BIOSCIENCES CORPORATION (US) 2011-12-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130310357-A1 Azolyl Urea Compounds and Methods of Use Thereof CSF1R, CSF3R, ARG1 FLT3 4/4885CSF1R 1/4885PDGFRB 733/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.