SCHEMBL1699170

SCHEMBL1699170

O=c1[nH]c2cc(CCCl)cnc2n1-c1ccc(O)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
MAP3K11 Q16584 7/20 0.39
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
PABPC1 P11940 1/20 0.36
KMT2A Q03164 1/20 0.36
MTOR P42345 2/20 0.34
KCNH2 Q12809 1/20 0.33
DAO P14920 1/20 0.33
GSK3B P49841 1/20 0.32
HSP90AA1 P07900 2/20 0.32
PDE4B Q07343 1/20 0.32
TDP2 O95551 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699176 0.83 NPC1 (0.49) MEN1KMT2ATDP2
SCHEMBL1699133 0.71 DAO (0.58) ESR1ESR2MAP3K11DAOHSP90AA1
SCHEMBL1699169 0.66 MAP3K11 (0.39) ESR1ESR2MAP3K11MEN1LMNA
SCHEMBL9981622 0.65 NPC1 (0.58) MEN1KMT2ATDP2
SCHEMBL725715 0.65 MAP3K11 (0.48) ESR1ESR2MAP3K11MEN1KMT2A
SCHEMBL15427058 0.65 KCNH2 (0.73) MEN1LMNAPABPC1KMT2AKCNH2
SCHEMBL1699212 0.65 MAP3K11 (0.40) ESR1ESR2MAP3K11MEN1LMNA
SCHEMBL1699188 0.65 NPC1 (0.48) KMT2AKCNH2TDP2
SCHEMBL1565665 0.64 MEN1 (0.44) MAP3K11MEN1LMNAPABPC1KMT2A
SCHEMBL1699264 0.64 MAP3K11 (0.40) ESR1ESR2MAP3K11MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed