SCHEMBL1699212

SCHEMBL1699212

CCc1cnc2c([nH]c(=O)n2-c2ccc(O)cc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 6/20 0.40
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
KDM4E B2RXH2 4/20 0.37
GAA P10253 2/20 0.37
HSD17B10 Q99714 2/20 0.37
MAPK1 P28482 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
RXFP1 Q9HBX9 2/20 0.35
GRM1 Q13255 1/20 0.34
CSNK2A1 P68400 1/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
HSP90AA1 P07900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699264 0.84 MAP3K11 (0.40) MAP3K11ESR1ESR2KDM4EGAA
SCHEMBL1699349 0.83 MAP3K11 (0.38) MAP3K11ESR1ESR2KDM4EGAA
SCHEMBL1699242 0.82 L3MBTL1 (0.56) KDM4EGAAALDH1A1CSNK2A1TSHR
SCHEMBL1699077 0.82 MAP3K11 (0.39) MAP3K11ESR1ESR2KDM4EGAA
SCHEMBL1699291 0.80 HSP90AA1 (0.40) KDM4EGAAHSD17B10ALDH1A1HPGD
SCHEMBL1699169 0.80 MAP3K11 (0.39) MAP3K11ESR1ESR2KDM4EGAA
SCHEMBL15385957 0.76 MAP3K11 (0.41) MAP3K11ESR1ESR2KDM4EGAA
SCHEMBL1699098 0.73 DRD1 (0.44) MEN1KMT2ALMNA
SCHEMBL1699258 0.67 L3MBTL1 (0.55) ALDH1A1CSNK2A1LMNATSHR
SCHEMBL1699284 0.67 MAP3K11 (0.39) MAP3K11ESR1ESR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed