SCHEMBL1699258

SCHEMBL1699258

Cc1c(C(C)C)cnc2c1[nH]c(=O)n2-c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.55
NPC1 O15118 2/20 0.55
RAB9A P51151 2/20 0.55
PKM P14618 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
NOX4 Q9NPH5 1/20 0.40
TDP2 O95551 1/20 0.40
CSNK2A2 P19784 1/20 0.40
CSNK2B P67870 1/20 0.40
CSNK2A1 P68400 1/20 0.40
MCHR1 Q99705 2/20 0.39
KCNH2 Q12809 1/20 0.39
BCL2 P10415 1/20 0.39
MDM2 Q00987 1/20 0.39
MCL1 Q07820 1/20 0.39
LMNA P02545 1/20 0.38
PIK3CA P42336 1/20 0.38
PRKDC P78527 1/20 0.38
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699242 0.86 L3MBTL1 (0.56) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699185 0.84 NPC1 (0.50) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699310 0.81 NPC1 (0.59) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699528 0.78 NPC1 (0.51) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699174 0.78 NPC1 (0.51) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699265 0.78 NPC1 (0.46) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL9981622 0.78 NPC1 (0.58) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699188 0.74 NPC1 (0.48) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699315 0.74 NPC1 (0.50) L3MBTL1NPC1RAB9APKMSMN1; SMN2
SCHEMBL1699125 0.72 NPC1 (0.56) L3MBTL1NPC1RAB9APKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed