SCHEMBL1699185

SCHEMBL1699185

CC(C)c1c(Cl)cnc2c1[nH]c(=O)n2-c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
BCL2 P10415 1/20 0.39
MDM2 Q00987 1/20 0.39
MCL1 Q07820 1/20 0.39
CSNK2A2 P19784 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
KCNH2 Q12809 1/20 0.38
MCHR1 Q99705 1/20 0.38
PRMT5 O14744 2/20 0.38
EGFR P00533 1/20 0.38
TDP2 O95551 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
PPARG P37231 1/20 0.37
NCOA2 Q15596 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699234 0.89 L3MBTL1 (0.54) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699174 0.85 NPC1 (0.51) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699258 0.84 L3MBTL1 (0.55) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699242 0.78 L3MBTL1 (0.56) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699528 0.77 NPC1 (0.51) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699310 0.77 NPC1 (0.59) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699188 0.77 NPC1 (0.48) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL9981622 0.76 NPC1 (0.58) NPC1RAB9AL3MBTL1PKMSMN1; SMN2
SCHEMBL1699476 0.74 PDE10A (0.36)
SCHEMBL1699176 0.73 NPC1 (0.49) NPC1RAB9AL3MBTL1PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed