SCHEMBL17004199

SCHEMBL17004199

c1cnn(-c2cncc(OC3C4CC5CC3CN(C5)C4)c2)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
NOTUM Q6P988 1/20 0.32
HSD11B1 P28845 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31
HCRTR1 O43613 3/20 0.31
HCRTR2 O43614 3/20 0.31
HRH3 Q9Y5N1 2/20 0.31
DGAT2 Q96PD7 1/20 0.30
MAPK1 P28482 1/20 0.30
ICAM1 P05362 1/20 0.30
SELE P16581 1/20 0.30
VCAM1 P19320 1/20 0.30
KCNH2 Q12809 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825645 0.76 CHRNB2 (0.41) CHRNB2CHRNA4
SCHEMBL17004288 0.76 FLT3 (0.34) CHRNB2CHRNA4
SCHEMBL17004290 0.75 CHRNB2 (0.40) CHRNB2CHRNA4
SCHEMBL17004272 0.75 CHRNB2 (0.40) KDM4ECHRNB2CHRNA4
SCHEMBL17004218 0.75 CHRNB2 (0.42) CHRNB2CHRNA4
SCHEMBL17004197 0.72
SCHEMBL3829106 0.71 OPRK1 (0.48) SIRT2SIRT1SIRT3CHRNB2CHRNA4
SCHEMBL17004327 0.71 MKNK1 (0.40) CHRNB2CHRNA4
SCHEMBL24921171 0.70 KDM4E (0.44) KDM4EALDH1A1NOTUMCHRNB2CHRNA4
SCHEMBL17004225 0.68 CHRNB2 (0.32) CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed