SCHEMBL17004265

SCHEMBL17004265

c1ccc(-c2ccc(OC3C4CC5CC3CN(C5)C4)nc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.40
CHRNA7 P36544 4/20 0.37
KCNH2 Q12809 3/20 0.37
KDR P35968 2/20 0.36
CHRNB2 P17787 3/20 0.35
CHRNB4 P30926 3/20 0.35
CHRNA3 P32297 3/20 0.35
CHRNA4 P43681 3/20 0.35
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
OPRK1 P41145 1/20 0.33
ATM Q13315 1/20 0.33
NAAA Q02083 1/20 0.33
MCHR1 Q99705 1/20 0.33
USP30 Q70CQ3 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
RET P07949 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004245 0.89 CHRNB4 (0.43) FAAHCHRNA7KCNH2CHRNB2CHRNB4
SCHEMBL17004220 0.88 CHRNB2 (0.36) FAAHCHRNA7CHRNB2CHRNB4CHRNA3
SCHEMBL17004293 0.86 CHRNB2 (0.34) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004269 0.84 CHRNB2 (0.35) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL17004292 0.83 MAOB (0.33) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL17004216 0.83 HCRTR1 (0.30) FAAHHCRTR1HCRTR2RET
SCHEMBL17004214 0.80 HCRTR2 (0.39) HCRTR1HCRTR2
SCHEMBL17004185 0.80 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL17004198 0.79 FURIN (0.40) HCRTR1HCRTR2NAAARET
SCHEMBL17004324 0.79 CHRNA7 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed