SCHEMBL17004292

SCHEMBL17004292

c1csc(-c2ccc(OC3C4CC5CC3CN(C5)C4)nc2)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
EGLN1 Q9GZT9 1/20 0.33
FLT3 P36888 2/20 0.33
NEK2 P51955 1/20 0.33
CHEK1 O14757 1/20 0.33
CHEK2 O96017 1/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
CYP17A1 P05093 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
CYP2E1 P05181 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2A6 P11509 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2B6 P20813 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004265 0.83 FAAH (0.40) KCNH2HCRTR1HCRTR2CHRNB2CHRNB4
SCHEMBL17004220 0.81 CHRNB2 (0.36) FLT3CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL17004245 0.80 CHRNB4 (0.43) ALDH1A1CYP3A4CYP2A6KCNH2CHRNB2
SCHEMBL17004293 0.79 CHRNB2 (0.34) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL17004239 0.79 CHRNA7 (0.47) KCNH2CHRNB2CHRNB4CHRNA3CHRNA7
SCHEMBL17004269 0.77 CHRNB2 (0.35) CHEK1CHEK2KCNH2HRH3HCRTR1
SCHEMBL17004214 0.76 HCRTR2 (0.39) HCRTR1HCRTR2
SCHEMBL17004185 0.76 HCRTR1 (0.39) HCRTR1HCRTR2
SCHEMBL17004198 0.72 FURIN (0.40) FLT3CYP3A4HCRTR1HCRTR2
SCHEMBL17004212 0.72 CHRNA7 (0.56) KCNH2CHRNB2CHRNB4CHRNA3CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed