SCHEMBL17008294

SCHEMBL17008294

COC(=O)C1CC(F)CCC1c1nn(-c2ccc(F)cn2)cc1-c1ccc(N2CCS(=O)(=O)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 9/20 0.51
ALDH1A1 P00352 1/20 0.34
SLC6A9 P48067 6/20 0.34
GPR119 Q8TDV5 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVR1 Q04771 1/20 0.33
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18279761 1.00 CTSK (0.51) CTSKALDH1A1SLC6A9GPR119TGFBR1
SCHEMBL17008292 0.94 CTSK (0.45) CTSKGPR119
SCHEMBL17008214 0.91 CTSK (0.52) CTSKSLC6A9GPR119FAAH
SCHEMBL18279702 0.91 CTSK (0.52) CTSKSLC6A9GPR119FAAH
SCHEMBL18279805 0.85 CTSK (0.71) CTSK
SCHEMBL17008308 0.85 CTSK (0.71) CTSK
SCHEMBL18279806 0.85 CTSK (0.71) CTSK
SCHEMBL17008212 0.85 CTSK (0.45) CTSKSLC6A9GPR119
SCHEMBL18279701 0.85 CTSK (0.45) CTSKSLC6A9GPR119
SCHEMBL18279712 0.84 CTSK (0.46) CTSKALDH1A1SLC6A9TGFBR1ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015120580-A1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-08-20 WO disclosed