SCHEMBL17009229

SCHEMBL17009229

C[C@@H]1CCCN[C@@H]1CNc1nccc(Cl)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.42
HRH4 Q9H3N8 3/20 0.38
PAK4 O96013 2/20 0.36
PAK1 Q13153 2/20 0.36
CHRNA3 P32297 2/20 0.34
PRPS1 P60891 1/20 0.34
GNRHR P30968 1/20 0.33
CDC7 O00311 2/20 0.33
ROCK2 O75116 1/20 0.33
CCNB2 O95067 1/20 0.33
MAP4K4 O95819 1/20 0.33
CDK1 P06493 1/20 0.33
RET P07949 1/20 0.33
CCNB1 P14635 1/20 0.33
PRKACA P17612 1/20 0.33
CDK2 P24941 1/20 0.33
GSK3B P49841 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
HIPK2 Q9H2X6 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17009227 1.00 HCRTR1 (0.42) HCRTR1HRH4PAK4PAK1CHRNA3
SCHEMBL15174141 0.79 HCRTR1 (0.39) HCRTR1CHRNA3
SCHEMBL16277337 0.79 HCRTR1 (0.39) HCRTR1CHRNA3
SCHEMBL2578413 0.73 HRH4 (0.55) HRH4PAK4PAK1GNRHRCDC7
SCHEMBL22761650 0.73 HCRTR1 (0.39) HCRTR1HRH3
SCHEMBL17009213 0.71 PRPS1 (0.36) HCRTR1PRPS1CDK1CDK2
SCHEMBL16277755 0.68 HCRTR1 (0.47) HCRTR1
SCHEMBL18734332 0.68 HCRTR1 (0.47) HCRTR1
SCHEMBL16284061 0.67 HCRTR1 (0.33) HCRTR1IRAK4HRH3
SCHEMBL1519442 0.66 LMNA (0.47) HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015123355-A1 SUBSTITUTED PROLINES / PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS EOLAS THERAPEUTICS, INC. (US) 2015-08-20 WO disclosed