SCHEMBL17009402

SCHEMBL17009402

Cc1ccc(-c2ccc(C(F)(F)F)cn2)c(C=O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.46
FEN1 P39748 1/20 0.46
HCRTR1 O43613 3/20 0.39
HCRTR2 O43614 1/20 0.39
KDM4E B2RXH2 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KIF11 P52732 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
PDE2A O00408 1/20 0.36
ALDH1A1 P00352 1/20 0.36
PKM P14618 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMO Q99835 1/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18752609 0.78 KDM4E (0.41) HCRTR1HCRTR2KDM4ENPSR1LMNA
SCHEMBL16277360 0.77 DHODH (0.51) ALOX5APFEN1HCRTR1HCRTR2KDM4E
SCHEMBL19248537 0.76 CYP1A2 (0.56) ALOX5APFEN1KDM4ENPSR1KIF11
SCHEMBL30540196 0.74 ALOX5AP (0.39) ALOX5APFEN1KDM4ELMNAALDH1A1
SCHEMBL26635201 0.74 ALOX5AP (0.39) ALOX5APFEN1KDM4ELMNAALDH1A1
SCHEMBL3102205 0.74 KDM4E (0.42) ALOX5APFEN1KDM4ENPSR1LMNA
SCHEMBL24689583 0.73 CCR1 (0.64) KDM4ENPSR1SMN1; SMN2KIF11CYP1A2
SCHEMBL28862771 0.73 FEN1 (0.46) ALOX5APFEN1NPSR1LMNAKIF11
SCHEMBL18003550 0.72 KIF11 (0.42) ALOX5APFEN1KDM4ENPSR1SMN1; SMN2
SCHEMBL16278041 0.72 NPC1 (0.47) KDM4ENPSR1LMNAHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015123355-A1 SUBSTITUTED PROLINES / PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS EOLAS THERAPEUTICS, INC. (US) 2015-08-20 WO disclosed