SCHEMBL1701031

SCHEMBL1701031

Fc1[c]ccc(-c2ccc(-c3cc4c(cc3Cl)CCO4)cn2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 2/20 0.38
PRKAG1 P54619 2/20 0.38
PRKAA2 P54646 2/20 0.38
PRKAA1 Q13131 2/20 0.38
PRKAG3 Q9UGI9 2/20 0.38
PRKAG2 Q9UGJ0 2/20 0.38
PRKAB1 Q9Y478 2/20 0.38
FABP4 P15090 5/20 0.33
STIM1 Q13586 4/20 0.33
ORAI1 Q96D31 4/20 0.33
RAB9A P51151 3/20 0.33
MAPT P10636 2/20 0.33
DYRK1A Q13627 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NPC1 O15118 2/20 0.31
FABP3 P05413 1/20 0.31
PLA2G10 O15496 1/20 0.30
ERN1 O75460 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1701271 0.74 DYRK1A (0.46) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL1701329 0.69 DYRK1A (0.46) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL18952827 0.69 BACE1 (0.40) RAB9ASMN1; SMN2NPC1
SCHEMBL14225980 0.68 STIM1 (0.55) STIM1ORAI1MAPTNPC1
SCHEMBL12155600 0.67 STIM1 (0.41) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL12156240 0.67 STIM1 (0.47) FABP4STIM1ORAI1RAB9ASMN1; SMN2
SCHEMBL1701214 0.67 STIM1 (0.38) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL2546978 0.67 SMN1; SMN2 (0.54) STIM1ORAI1RAB9AMAPTSMN1; SMN2
SCHEMBL11490989 0.67 PRKAB2 (0.45) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL3822351 0.66 GRM5 (0.38) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563776-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2011139489-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-11-10 WO disclosed