SCHEMBL17012016

SCHEMBL17012016

CC(C)NC(=O)c1cccc(C(O)NCc2cccc(Cl)c2)n1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.45
SLC2A1 P11166 1/20 0.43
ALDH1A1 P00352 2/20 0.40
MEN1 O00255 1/20 0.40
HCRTR1 O43613 1/20 0.40
KMT2A Q03164 1/20 0.40
HPGD P15428 1/20 0.40
BRD4 O60885 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CNR2 P34972 3/20 0.39
APEX1 P27695 1/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NPC1 O15118 1/20 0.39
CNR1 P21554 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8205783 0.82 MEN1 (0.52) POLBSLC2A1ALDH1A1MEN1HCRTR1
SCHEMBL21776043 0.73 HPGD (0.60) ALDH1A1KMT2AHPGD
SCHEMBL9415944 0.73 PNMT (0.53) SLC2A1
SCHEMBL25820326 0.72 CNR1 (0.46) ALDH1A1MEN1KMT2AKDM4ECNR2
SCHEMBL30471855 0.70 PNMT (0.56) SLC2A1
SCHEMBL12000668 0.70 PNMT (0.56) SLC2A1
SCHEMBL8198502 0.70 SMN1; SMN2 (0.53) ALDH1A1MEN1KMT2AHPGDKDM4E
SCHEMBL28386072 0.69 CTSA (0.54) POLBALDH1A1MEN1KMT2AKDM4E
SCHEMBL8198970 0.68 ROCK2 (0.48) ALDH1A1MEN1KMT2AHPGDBRD4
SCHEMBL12853358 0.68 HPGD (0.53) POLBALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2132178-B1 JNK INHIBITORS MERCK SHARP & DOHME (US) 2015-08-19 EP disclosed