SCHEMBL17023181

SCHEMBL17023181

CCN1CCN(c2ccc(NC(=O)Oc3ccc(-c4c(Cl)c(OC)cc(OC)c4Cl)c4cccnc34)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FGFR3 P22607 16/20 0.59
FGFR1 P11362 5/20 0.50
FGFR2 P21802 4/20 0.50
FGFR4 P22455 4/20 0.50
JAK2 O60674 2/20 0.48
ABL1 P00519 2/20 0.48
INSR P06213 2/20 0.48
LCK P06239 2/20 0.48
FYN P06241 2/20 0.48
YES1 P07947 2/20 0.48
LYN P07948 2/20 0.48
RET P07949 2/20 0.48
MET P08581 2/20 0.48
ROS1 P08922 2/20 0.48
KIT P10721 2/20 0.48
SRC P12931 2/20 0.48
BRAF P15056 2/20 0.48
PDGFRA P16234 2/20 0.48
FLT1 P17948 2/20 0.48
TYK2 P29597 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17023062 0.91 FGFR3 (0.66) FGFR3FGFR1FGFR2FGFR4JAK2
SCHEMBL12678403 0.88 FGFR3 (0.71) FGFR3FGFR1FGFR2FGFR4NR4A1
SCHEMBL17023033 0.87 FGFR3 (0.58) FGFR3
SCHEMBL17023176 0.84 FGFR3 (0.80) FGFR3FGFR1FGFR2FGFR4JAK2
SCHEMBL17023113 0.82 FGFR3 (0.68) FGFR3
SCHEMBL17023067 0.82 FGFR3 (0.65) FGFR3
SCHEMBL17023154 0.82 FGFR3 (0.65) FGFR3FGFR1KDRPOLB
SCHEMBL1126632 0.81 FGFR3 (0.83) FGFR3
SCHEMBL17023160 0.81 FGFR3 (0.80) FGFR3
SCHEMBL17023178 0.81 FGFR3 (0.58) FGFR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282995-B1 DERIVATIVES OF QUINOLINES AND QUINOXALINES AS PROTEIN TYROSINE KINASE INHIBITORS NOVARTIS AG (CH) 2015-08-26 EP claimed